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DRUG CLASS:
ERK1 inhibitor
DRUG CLASS:
ERK1 inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
BVD-523 (17)
ERAS-007 (13)
JSI-1187 (4)
ASTX029 (4)
LTT462 (3)
LY3214996 (3)
AEZS 136 (1)
D3S-002 (0)
HH2710 (0)
MK-8353 (0)
ATG-017 (0)
BVD-523 (17)
ERAS-007 (13)
JSI-1187 (4)
ASTX029 (4)
LTT462 (3)
LY3214996 (3)
AEZS 136 (1)
D3S-002 (0)
HH2710 (0)
MK-8353 (0)
ATG-017 (0)
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Associations
(46)
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Trials
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BRAF L597Q
Solid Tumor
BRAF L597Q
Solid Tumor
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BRAF G469A
Solid Tumor
BRAF G469A
Solid Tumor
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BRAF G469V
Solid Tumor
BRAF G469V
Solid Tumor
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BRAF L485W
Solid Tumor
BRAF L485W
Solid Tumor
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BVD-523
Sensitive: B - Late Trials
BVD-523
Sensitive
:
B
BRAF V600E
Melanoma
BRAF V600E
Melanoma
JSI-1187
Sensitive: C2 – Inclusion Criteria
JSI-1187
Sensitive
:
C2
JSI-1187
Sensitive: C2 – Inclusion Criteria
JSI-1187
Sensitive
:
C2
NRAS mutation
Melanoma
NRAS mutation
Melanoma
BVD-523
Sensitive: C2 – Inclusion Criteria
BVD-523
Sensitive
:
C2
BVD-523
Sensitive: C2 – Inclusion Criteria
BVD-523
Sensitive
:
C2
BRAF V600E
Colorectal Cancer
BRAF V600E
Colorectal Cancer
LY3214996
Sensitive: C2 – Inclusion Criteria
LY3214996
Sensitive
:
C2
LY3214996
Sensitive: C2 – Inclusion Criteria
LY3214996
Sensitive
:
C2
BRAF mutation
Melanoma
BRAF mutation
Melanoma
BVD-523
Sensitive: C2 – Inclusion Criteria
BVD-523
Sensitive
:
C2
BVD-523
Sensitive: C2 – Inclusion Criteria
BVD-523
Sensitive
:
C2
KRAS mutation
Colorectal Cancer
KRAS mutation
Colorectal Cancer
ERAS-007
Sensitive: C2 – Inclusion Criteria
ERAS-007
Sensitive
:
C2
ERAS-007
Sensitive: C2 – Inclusion Criteria
ERAS-007
Sensitive
:
C2
BRAF V600E
Colorectal Cancer
BRAF V600E
Colorectal Cancer
ERAS-007
Sensitive: C2 – Inclusion Criteria
ERAS-007
Sensitive
:
C2
ERAS-007
Sensitive: C2 – Inclusion Criteria
ERAS-007
Sensitive
:
C2
KRAS mutation
Non Small Cell Lung Cancer
KRAS mutation
Non Small Cell Lung Cancer
ERAS-007 + ERAS-601
Sensitive: C2 – Inclusion Criteria
ERAS-007 + ERAS-601
Sensitive
:
C2
ERAS-007 + ERAS-601
Sensitive: C2 – Inclusion Criteria
ERAS-007 + ERAS-601
Sensitive
:
C2
BRAF V600E
Melanoma
BRAF V600E
Melanoma
LY3214996
Sensitive: C2 – Inclusion Criteria
LY3214996
Sensitive
:
C2
LY3214996
Sensitive: C2 – Inclusion Criteria
LY3214996
Sensitive
:
C2
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