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BIOMARKER:
PIK3R1 mutation
i
Other names:
PIK3R1, Phosphoinositide-3-Kinase Regulatory Subunit 1, Phosphatidylinositol 3-Kinase 85 KDa Regulatory Subunit Alpha, Phosphoinositide-3-Kinase, Regulatory Subunit 1 (Alpha), Phosphatidylinositol 3-Kinase Regulatory Subunit Alpha, Phosphoinositide-3-Kinase Regulatory Subunit Alpha, PtdIns-3-Kinase Regulatory Subunit Alpha, PI3K Regulatory Subunit Alpha, PI3-Kinase Subunit P85-Alpha, GRB1, Phosphatidylinositol 3-Kinase, Regulatory Subunit, Polypeptide 1 (P85 Alpha), Phosphatidylinositol 3-Kinase
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Entrez ID:
5295
Related biomarkers:
Expression
Mutation
Others
‹
PIK3R1 overexpression (2)
PIK3R1 overexpression (2)
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Associations
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VERI cancer hierarchy
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PIK3R1 mutation
Hormone Receptor Positive Breast Cancer
PIK3R1 mutation
Hormone Receptor Positive Breast Cancer
lenvatinib
Resistant: C3 – Early Trials
lenvatinib
Resistant
:
C3
lenvatinib
Resistant: C3 – Early Trials
lenvatinib
Resistant
:
C3
PIK3R1 mutation
Endometrial Cancer
PIK3R1 mutation
Endometrial Cancer
LY3023414
Sensitive: C3 – Early Trials
LY3023414
Sensitive
:
C3
LY3023414
Sensitive: C3 – Early Trials
LY3023414
Sensitive
:
C3
PIK3R1 mutation
Breast Cancer
PIK3R1 mutation
Breast Cancer
alpelisib + L-NMMA
Sensitive: D – Preclinical
alpelisib + L-NMMA
Sensitive
:
D
alpelisib + L-NMMA
Sensitive: D – Preclinical
alpelisib + L-NMMA
Sensitive
:
D
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