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DRUG CLASS:
Src kinase inhibitor
DRUG CLASS:
Src kinase inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
dasatinib (215)
bosutinib (46)
TPX-0022 (8)
AZD0530 (7)
BAL3833 (4)
NXP900 (3)
PP2 (2)
TPX-0046 (2)
AZD 0424 (0)
JNJ-26483327 (0)
tirbanibulin ointment (0)
XL228 (0)
KX-01 oral (0)
dasatinib (215)
bosutinib (46)
TPX-0022 (8)
AZD0530 (7)
BAL3833 (4)
NXP900 (3)
PP2 (2)
TPX-0046 (2)
AZD 0424 (0)
JNJ-26483327 (0)
tirbanibulin ointment (0)
XL228 (0)
KX-01 oral (0)
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Associations
(288)
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BCR-ABL1 fusion
Chronic Myeloid Leukemia
BCR-ABL1 fusion
Chronic Myeloid Leukemia
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
BCR-ABL1 fusion
Acute Lymphocytic Leukemia
BCR-ABL1 fusion
Acute Lymphocytic Leukemia
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
BCR-ABL1 fusion
Chronic Myeloid Leukemia
BCR-ABL1 fusion
Chronic Myeloid Leukemia
bosutinib
Sensitive: A1 - Approval
bosutinib
Sensitive
:
A1
bosutinib
Sensitive: A1 - Approval
bosutinib
Sensitive
:
A1
BCR-ABL1 fusion
B Acute Lymphoblastic Leukemia
BCR-ABL1 fusion
B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
BCR-ABL1 V299L
Acute Lymphocytic Leukemia
BCR-ABL1 V299L
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317I
Acute Lymphocytic Leukemia
BCR-ABL1 F317I
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 V299L
Chronic Myeloid Leukemia
BCR-ABL1 V299L
Chronic Myeloid Leukemia
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
BCR-ABL1 T315I
Chronic Myeloid Leukemia
BCR-ABL1 T315I
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315I
Chronic Myeloid Leukemia
BCR-ABL1 T315I
Chronic Myeloid Leukemia
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
bosutinib
Resistant: A2 - Guideline
bosutinib
Resistant
:
A2
No biomarker
Chronic Myeloid Leukemia
No biomarker
Chronic Myeloid Leukemia
bosutinib
Sensitive: A2 - Guideline
bosutinib
Sensitive
:
A2
bosutinib
Sensitive: A2 - Guideline
bosutinib
Sensitive
:
A2
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