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DRUG CLASS:
CDK2 inhibitor
DRUG CLASS:
CDK2 inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
BLU-222 (4)
INX-315 (2)
PF-07104091 (1)
AVZO-021 (0)
FN-1501 (0)
GW8510 (0)
RLY-2139 (0)
BLU-222 (4)
INX-315 (2)
PF-07104091 (1)
AVZO-021 (0)
FN-1501 (0)
GW8510 (0)
RLY-2139 (0)
›
Associations
(8)
News
Trials
VERI cancer hierarchy
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CCNE1 amplification
Ovarian Cancer
CCNE1 amplification
Ovarian Cancer
BLU-222
Sensitive: C2 – Inclusion Criteria
BLU-222
Sensitive
:
C2
BLU-222
Sensitive: C2 – Inclusion Criteria
BLU-222
Sensitive
:
C2
CCNE1 amplification
Ovarian Cancer
CCNE1 amplification
Ovarian Cancer
INX-315
Sensitive: C2 – Inclusion Criteria
INX-315
Sensitive
:
C2
INX-315
Sensitive: C2 – Inclusion Criteria
INX-315
Sensitive
:
C2
HR positive
HER2 Negative Breast Cancer
HR positive
HER2 Negative Breast Cancer
PF-07104091
Sensitive: C2 – Inclusion Criteria
PF-07104091
Sensitive
:
C2
PF-07104091
Sensitive: C2 – Inclusion Criteria
PF-07104091
Sensitive
:
C2
HR positive
HER2 Negative Breast Cancer
HR positive
HER2 Negative Breast Cancer
BLU-222
Sensitive: C3 – Early Trials
BLU-222
Sensitive
:
C3
BLU-222
Sensitive: C3 – Early Trials
BLU-222
Sensitive
:
C3
CCNE1 amplification
Breast Cancer
CCNE1 amplification
Breast Cancer
CDK2 inhibitor
Sensitive: D – Preclinical
CDK2 inhibitor
Sensitive
:
D
CDK2 inhibitor
Sensitive: D – Preclinical
CDK2 inhibitor
Sensitive
:
D
HR positive
HER2 Negative Breast Cancer
HR positive
HER2 Negative Breast Cancer
ribociclib + BLU-222
Sensitive: D – Preclinical
ribociclib + BLU-222
Sensitive
:
D
ribociclib + BLU-222
Sensitive: D – Preclinical
ribociclib + BLU-222
Sensitive
:
D
CCNE1 amplification
Gastric Cancer
CCNE1 amplification
Gastric Cancer
INX-315
Sensitive: D – Preclinical
INX-315
Sensitive
:
D
INX-315
Sensitive: D – Preclinical
INX-315
Sensitive
:
D
HR positive
HER2 Negative Breast Cancer
HR positive
HER2 Negative Breast Cancer
palbociclib + BLU-222
Sensitive: D – Preclinical
palbociclib + BLU-222
Sensitive
:
D
palbociclib + BLU-222
Sensitive: D – Preclinical
palbociclib + BLU-222
Sensitive
:
D
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